Introduction to Desipramine


[​IMG]

Pharmacology of Desipramine

LD50 (mg/kg) :
Mice : 500 (orally), 94 (intraperitoneally), 420 (sub cutaneously)
Rat : 385 (orally), 48 (intraperitoneally), 183 (sub cutaneously)

Chemistry of Desipramine

Column 1 Column 2
Systematic (IUPAC) name: 10,11-Dihydro-N-methyl-5H-dibenz[b,f]azepine-5-propanamine
Synonyms: 10,11-dihydro-5-[3-(methylamino)propyl]-5H-dibenz[b,f]azepine, 5-([gamma]-methylaminopropyl)-iminodibenzyl, N-(3-methylaminopropyl)iminodibenzyl, desmethylimipramine, norimipramine; G-35020, JB-8181, NSC-114901, Norpramin, Nortimil, Pertofran, Pertofrane, Petylyl (hydrochloride)
Molecular Formula: C18H22N2
Molar mass: 266.39 g/mol, 302.85 g/mol (hydrochloride)
CAS Registry Number: 50-47-5, 58-28-6 (hydrochloride)
Melting Point: 215-216°C (hydrochloride)
Boiling Point: 172-174°C @ 0.02 mmHg
Flash Point: no data
Solubility: Freely soluble in methanol, chloroform. Soluble in water, alcohol. Insoluble in ether.
Additionnal data: none
Notes: White to off white crystals from methanol
[1]

References


[1]Merck Index, fifteenth edition (2013)

This page has been seen 11,557 times.